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APIs thiab Intermediates
Fruquintinib CAS 1194506-26-7

Fruquintinib CAS 1194506-26-7

CAS NO: 1194506-26-7
Cov roj formula: C21H19N3O5
Molecular Luj: 393.39
EINECS NO: 962-485-3
MDL NO: N/A

Txhawb tshuaj

Product Description:

Khoom npe: fruquintinib CAS 1194506-26-7

 

Synonyms:

6-(6,7-dimethoxyquinazolin-4-}yl)oxy-N,2-dimethyl-1-benzofuran-3-carboxamide;

 

Chemical & Physical Properties:

Cov tsos mob: dawb mus rau cov hmoov dawb dawb

Assay: Ntau dua lossis sib npaug rau 99.0%

Kub taw tes: 600.5 degree (Predicted)

Qhov ceev: 1.302g / cm3

Solubility: Soluble hauv DMSO (txog 5 mg / ml).

 

 

Siv

Fruquintinib (HMPL-013) yog ib qho kev xaiv VEGFR-1/2/3 tyrosine kinase inhibitor. Nws tau pom zoo los ntawm FDA thaum Lub Kaum Ib Hlis 8, 2023 rau kev kho mob ntawm cov neeg laus uas muaj mob qog nqaij hlav hauv plab hnyuv loj. thiab cov neeg mob no yav dhau los tau txais fluoropyrimidine, oxaliplatin thiab irinotecan chemotherapy, anti-vascular endothelial txoj kev loj hlob zoo tshaj plaws, thiab anti-epidermal growth factor receptor (EGFR) kho. Fruquintinib kuj tau pom tias txhim kho kev paub tsis txaus ntseeg thiab kev hloov pauv pathological hauv tus qauv nas ntawm cerebral amyloid angiopathy (CAA).

 

Yog tias koj txaus siab rau peb cov khoom lossis muaj lus nug, thov koj xav tiv tauj peb!

 

Cov khoom raws li patent yog muab rau R & D lub hom phiaj nkaus xwb. Txawm li cas los xij, lub luag haujlwm kawg tsuas yog nrog tus neeg yuav khoom.

Cim npe nrov: fruquintinib cas 1194506-26-7, manufacturers, lwm tus neeg, Hoobkas, yuav, Tshuag

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