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Ntxiv:1002, Huanmao Tsev, No.105, Mengcheng Txoj kev, Hefei Lub zos, 230061 Tuam Tshoj
CAS TSIS TAU: 1207293-36-4
Cov mis mos molecular: C29H28N4O2
Molecular phaus: 464.55800
EINECS NO: Tsis yog
MDL NO: NA
Khoom Piav Qhia:
Khoom Lub Npe: BI-847325 CAS TSIS TAU: 1207293-36-4
Lub ntsiab lus:
3- [3-[[4-[(Dimethylamino) methyl] phenyl] amino] phenylmethylene] -2,3-dihydro-2-oxo-1H-indol-6-yl] -N-ethyl-2-propynamide;
Tshuaj& Lub Cev Muaj Zog:
Tshwm sim: Crystalline khoom
Kev Ntsuas: ≥98.0%
Ceev: 1.3 ± 0.1 g/cm3
Index ntawm Refraction: 1.673
Cia: 3 xyoos -20 ℃ hmoov; 6 lub hlis -80 ℃ hauv qhov hnyav.
BI-847325 yog qhov muaj nyob hauv qhov ncauj, thiab xaiv ob lub MEK/Aurora kinase inhibitor nrog IC50 ntawm 3 nM, 25 nM, 15 nM, 25 nM, thiab 4 nM rau Xenopus laevis Aurora B, tib neeg Aurora A thiab Aurora C, ntxiv rau tib neeg MEK1 thiab MEK2, feem.
Yog tias koj txaus siab rau peb cov khoom lossis muaj lus nug, thov koj xav tiv tauj peb!
Cov khoom lag luam nyob rau hauv patent tau muab rau R& D lub hom phiaj nkaus xwb. Txawm li cas los xij, lub luag haujlwm zaum kawg tshwj xeeb tshaj yog nrog tus neeg yuav khoom.
Cim npe nrov: bi-847325 cas 1207293-36-4, tuam ntxhab, cov chaw muag khoom, lub Hoobkas, yuav, hauv Tshuag