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CAS TSIS TAU: 417716-92-8
Cov Qauv Nqaij: C21H19ClN4O4
Cov Nqa Molecular: 426.85300
EINECS TSIS MUAJ: NA
MDL TSIS TAU: MFCD16038644
Khoom Qhia:
Khoom npe: lenvatinib CAS TSIS: 417716-92-8
Txhais:
E7080,E 7080;
Lenvatinib (E7080);
4- [3-chloro-4- (cyclopropylcarbamoylamino) phenoxy] -7-methoxyquinoline-6-carboxamide;
Tshuaj& Cov Khoom Uas Lub Cev:
Zog: Dawb kom dawb-tawm cov hmoov dawb dawb
Ntsuas: ≥98.0%
Qhov ceev: 1.469g / cm3
Lub Ntsiab Kub: 627.242 ℃ ntawm 760 mmHg
Flash Point: 333.144 ℃
Qhov Taw Qhia Txaus Nruab Nrab: 1.697
Solubility: Soluble hauv DMSO
Kev mob cia: Lub sijhawm luv cia (lub lis piam): 0 - 4 ℃ hauv qab qhuav; Lub sijhawm ntev cia (hli): -20 ℃ hauv qab qhuav
Cov Ntaub Ntawv Kev Nyab Xeeb:
Cov Kev Ceeb Toom Kom Raug Mob: Ua rau lub qhov muag mob siab heev. Xav tias tsam puas xeeb tub los sis tus menyuam hauv plab
Cov Lus Qhia Txog Kev Ceev Faj Dav: Ua kom tsis txhob ncav cuag cov menyuam.
Lenvatinib (lag luam npe Lenvima) yog ib hom tshuaj tiv thaiv qog noj ntshav rau kev kho qee yam mob qog noj ntshav, thiab muaj feem yuav ua rau lwm yam mob qog nqaij hlav thiab. Nws tau tsim los ntawm Eisai Co. thiab ua raws li ntau yam kinase inhibitor tiv thaiv VEGFR1, VEGFR2 thiab VEGFR3 kinases. E7080 (Lenvatinib) yog qhov sib txuam sib txuam ntawm VEGFR2 thiab VEGFR3 nrog IC50 ntawm 4 nM thiab 5.2 nM, ntsig txog.
Yog tias koj txaus siab rau peb cov khoom lossis muaj lus nug, thov koj xav tiv tauj peb!
Cov khoom lag luam hauv qab patent yog muab rau R& D lub hom phiaj nkaus xwb. Txawm li cas los xij, lub luag haujlwm kawg tau txiav txim siab nrog cov neeg yuav khoom.
Cim npe nrov: lenvatinib cas 417716-92-8, tuam ntxhab, lwm tus neeg, Hoobkas, yuav, hauv Tshuag