Hu rau:Errol Zhou (Mr.)
Tel: ntxiv 86-551-65523315
Mobile/WhatsApp: ntxiv 86 17705606359
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Email:sales@homesunshinepharma.com
Ntxiv:1002, Huanmao Tsev, No.105, Mengcheng Txoj kev, Hefei Lub zos, 230061 Tuam Tshoj
CAS TSIS TAU: 775351-65-0
Cov Qauv Nqaij: C6H13N5
Nqa Molecular: 155.20100
EINECS TSIS MUAJ: NA
MDL TSIS TAU: NA
Khoom Qhia:
Khoom npe: imeglimin CAS TSIS: 775351-65-0
Txhais:
Imeglimin;
UNII-UU226QGU97;
Tshuaj& Cov Khoom Uas Lub Cev:
Pom: Cov hmoov pob
Ntsuas: ≥98.0%
Qhov ceev: 1.29 ± 0.1 g / cm3 (Pom zoo)
Lub Ntsiab Kub: 239.9 ± 23.0 ℃ (Xav Tau)
Solubility: Soluble hauv DMSO
Imeglimin yog thawj zaug nyob rau hauv chav kawm tetrahydrotriazine tshiab uas muaj cov tshuaj tiv thaiv kab mob hauv lub qhov ncauj, cov glimins. Nws tau pom tias ua los ua rau lub siab, mob nqaij thiab pancreatic cells-cov cell mus rau qhov tsis tau tshwj xeeb ua rau cov tsis tseem ceeb ntawm hom ntshav qab zib hom 2. Imeglimin yog ib txoj kev sim tshuaj uas tau tsim los ua qhov ncauj tawm tsam ntshav qab zib. Nws yog ib qho oxidative phosphorylation blocker uas ua rau inhibit hepatic gluconeogenesis, ua rau cov leeg ua haujlwm ntau ntxiv, thiab rov qab muaj dej tsis muaj zog. Nws yuav yog thawj zaug ntawm chav kawm tshiab ntawm kev tiv thaiv ntshav qab zib yog tias nws pom zoo.
Imeglimin yog nyob rau hauv txoj kev loj hlob (ua tiav theem IIb kev soj ntsuam hauv tsev kho mob) rau siv ob qho tib si li monotherapy thiab hauv kev sib xyaw nrog lwm cov kev kho mob ntshav qab zib hom-2.
Ntau cov kev tshawb fawb raws tu qauv tau paub los ntawm ntau tus kws tshawb fawb. Cov kev tshawb pom thaum ntxov pom tias imeglimin muaj txiaj ntsig zoo li metformin hauv kev tswj hwm glycemic.
Yog tias koj txaus siab rau peb cov khoom lossis muaj lus nug, thov koj xav tiv tauj peb!
Cov khoom lag luam hauv qab patent yog muab rau R& D lub hom phiaj nkaus xwb. Txawm li cas los xij, lub luag haujlwm kawg tau txiav txim siab nrog cov neeg yuav khoom.
Cim npe nrov: imeglimin cas 775351-65-0, tuam ntxhab, lwm tus neeg, Hoobkas, yuav, hauv Tshuag