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CAS TSIS TAU: 872728-81-9
Cov Qauv Nqaij: C35H45N7O8S
Cov Nqa Molecular: 723.839
EINECS TSIS MUAJ: 828-727-6
MDL TSIS TAU: MFCD72728819
Khoom Qhia:
Khoom npe: Dabigatran Etexilate Mesylate CAS TSIS: 872728-81-9
Txhais:
Dabigatran etexilate methanesulfonate;
Ethyl N - [(2 - {[(4- {N - [(hexyloxy) carbonyl] carbamimidoyl} phenyl) amino] methyl} -1-methyl-1H-benzimidazol-5-yl) carbonyl] -N-2-pyridinyl -β-alaninate methanesulfonate (1: 1);
Tshuaj& Cov Khoom Uas Lub Cev:
Zog: Off-Dawb rau daj hmoov
Ntsuas: ≥99.0%
Dabigatran etexilate mesylate yog qhov tshuaj tiv thaiv thrombin tshwj xeeb uas siv hauv kev soj ntsuam thiab ib yam tshiab ntawm lub qhov ncauj tiv thaiv tsis tau. Nws cov tshuab ntawm kev ua yog inhibit qhov tsim ntawm fibrin los ntawm kev thim rov qab thiab muaj zog sib tw los khi rau cov fibrin kev khi qhov chaw ntawm thrombin, yog li inhibiting qhov tsim ntawm thrombus.
Dabigatran etexilate mesylate yog ib yam khoom ua los ntawm dabigatran, uas tau hloov pauv mus rau hauv cov dabigatran uas nquag ua tom qab lub cev hauv lub cev. Piv nrog warfarin, dabigatran etexilate mesylate tsis tas yuav saib xyuas kev sib xyaw ua ke thiab kev hloov kho thaum lub sijhawm kho, thiab tsis muaj kev cuam tshuam tsawg ntawm cov tshuaj thiab tsis cuam tshuam los ntawm kev noj, yog li txhim kho tus neeg mob' s kev ua raws kev noj tshuaj.
Txhua tus yuav tsum paub tias cov tshuaj warfarin tam sim no yog cov tshuaj tseem ceeb siv los tiv thaiv mob stroke thiab system embolism hauv cov neeg mob atrial fibrillation, thiab nws muaj qhov chaw tsis muaj peev xwm tiv thaiv kev kho mob ntawm cov neeg mob atrial fibrillation. Warfarin ib txwm raug suav hais tias yog kev kho mob antithrombotic hauv daim teb no. txuj ci kub. Txawm li cas los xij, hauv kev siv tshuaj, nws tau pom tias warfarin cuam tshuam nrog ntau yam tshuaj thiab kev noj haus, xws li quinolone thiab tshuaj tua kab mob macrolide. Nws yog feem ntau tsis tuaj yeem lees tias nws cov koob tshuaj yuav tsum tswj hwm nyob rau hauv kev kho lub qhov rai thiab muaj kev pheej hmoo los ntshav. Txhawm rau kom muaj kev nyab xeeb ntawm kev siv tshuaj, nws yog ib qho tsim nyog los soj ntsuam cov ntshav coagulation kev ua haujlwm thiab kho cov tshuaj ntau npaum li cas.
Dabigatran etexilate yog lwm qhov tshuaj tiv thaiv qhov ncauj tshiab uas tau pom zoo los ntawm Asmeskas Chaw Tswj Xyuas Khoom Noj thiab Tshuaj tom qab warfarin. Nws yog qhov tsis-peptide thrombin inhibitor uas tshwj xeeb thiab xaiv ua kom tsis txhob thrombin (Pub dawb los yog sib xyaw) kev ua haujlwm kom ua rau cov nyhuv anticoagulant. Nws tuaj yeem noj ntawm qhov ncauj, muaj hwj chim, tsis tas yuav tshuaj xyuas tshwj xeeb, thiab muaj kev sib txuam tshuaj tsawg dua. Nws yog qhov kev nce qib tseem ceeb hauv kev kho cov tshuaj tiv thaiv kab mob thiab kev ua kom muaj kev phom sij rau kev tiv thaiv kabmob, thiab nws yog qhov tseem ceeb. Tom qab lub qhov ncauj nqus tau los ntawm kev mob plab, nws tau hloov mus rau hauv dabigatran nrog kev cuam tshuam ncaj nraim hauv lub cev. Los ntawm kev khi rau cov fibrin tej chaw khi ntawm thrombin, nws tiv thaiv fibrinogen los ntawm kev zawm mus rau fibrin, yog li thaiv cov ntshav txhaws qhov kawg ntawm cov dej tsaws tsag network thiab thrombosis. Dabigatran tseem tuaj yeem cais tawm ntawm cov fibrin-thrombin conjugate thiab siv qhov ua rau lub ntsej muag tiv thaiv kev tsis haum.
Yog tias koj txaus siab rau peb cov khoom lossis muaj lus nug, thov hu rau peb!
Cov khoom lag luam hauv qab patent yog muab rau R& D lub hom phiaj nkaus xwb. Txawm li cas los xij, lub luag haujlwm kawg tau txiav txim siab nrog cov neeg yuav khoom.
Cim npe nrov: dabigatran etexilate mesylate cas 872728-81-9, tuam ntxhab, lwm tus neeg, Hoobkas, yuav, hauv Tshuag